SCHEMBL20170890

SCHEMBL20170890

CCc1cccnc1CNC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.40
SLC6A4 P31645 2/20 0.40
CYP2A6 P11509 1/20 0.40
SLC6A3 Q01959 1/20 0.40
TAAR1 Q96RJ0 2/20 0.38
HTR1A P08908 1/20 0.38
ADORA2A P29274 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35
KCNH2 Q12809 1/20 0.35
SCN5A Q14524 1/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
GABRA1 P14867 2/20 0.34
GABRB2 P47870 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
LMNA P02545 2/20 0.34
GPR84 Q9NQS5 1/20 0.34
ALOX15 P16050 1/20 0.34
SLC40A1 Q9NP59 1/20 0.34
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17667911 0.85 SLC6A2 (0.40) SLC6A2SLC6A4CYP2A6SLC6A3TAAR1
SCHEMBL13073821 0.82 ALDH1A1 (0.39) SLC6A2SLC6A4CYP2A6SLC6A3TAAR1
SCHEMBL242311 0.81 GABRA1 (0.41) TAAR1HTR1AALDH1A1KDM4EGABRA1
Ammonia Solution, Strong SCHEMBL25385979 0.79 GABRA1 (0.39) TAAR1HTR1AALDH1A1KDM4EGABRA1
SCHEMBL5786722 0.79 GABRA1 (0.39) TAAR1HTR1AALDH1A1KDM4EGABRA1
SCHEMBL27951839 0.79 HRH3 (0.42) SLC6A4CYP2A6TAAR1HRH3ALDH1A1
Hydrochloric Acid SCHEMBL28665184 0.78 GABRA1 (0.38) TAAR1HTR1AALDH1A1KDM4EGABRA1
SCHEMBL27939527 0.78 CYP2A6 (0.36) CYP2A6TAAR1HRH3ALDH1A1L3MBTL1
SCHEMBL5968788 0.78 HTR5A (0.37) ADORA2AALDH1A1KDM4ELMNAMAPT
Ammonia Solution, Strong SCHEMBL27939539 0.76 HTR2C (0.35) SLC6A4CYP2A6TAAR1HRH3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103570688-A 2,5-diaminomethylpyrazine compounds, drug compositions, preparation method and use thereof SHANGHAI INST MATERIA MEDICA 2014-02-12 CN claimed
WO-2023076237-A1 COMPOUNDS AS GLP-1R AGONISTS TERNS PHARMACEUTICALS, INC. (US) 2023-05-04 WO disclosed
EP-3038466-B1 2,2-DIFLUORODIOXOLO A2A RECEPTOR ANTAGONISTS MERCK SHARP & DOHME (US) 2018-05-23 EP disclosed
CN-103570688-A 2,5-diaminomethylpyrazine compounds, drug compositions, preparation method and use thereof SHANGHAI INST MATERIA MEDICA 2014-02-12 CN disclosed