SCHEMBL20171112

SCHEMBL20171112

CNSc1cccc(C)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 4/20 0.48
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
DDB1 Q16531 1/20 0.36
CRBN Q96SW2 1/20 0.36
TP53 P04637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
IDO1 P14902 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23048506 0.80 ACHE (0.46) ACHEALDH1A1MAPK1CYP1A2CYP3A4
SCHEMBL28492107 0.80 ACHE (0.46) ACHEALDH1A1MAPK1CYP1A2CYP3A4
SCHEMBL20902674 0.78 PTPN5 (0.37) CYP1A2CYP3A4MAPTCYP2C9CYP2C19
SCHEMBL20048798 0.76 TSHR (0.42) ALDH1A1MAPK1CYP1A2CYP3A4CYP2D6
SCHEMBL19222192 0.76 MAOA (0.46) ALDH1A1MAPK1MAPTNPSR1DDB1
SCHEMBL29468620 0.75 ACHE (0.58) ACHEALDH1A1MAPK1CYP1A2CYP3A4
SCHEMBL29468631 0.75 ACHE (0.58) ACHEALDH1A1MAPK1MAPTHTT
SCHEMBL576105 0.75 ACHE (0.58) ACHEALDH1A1MAPK1CYP1A2CYP3A4
SCHEMBL575896 0.75 ACHE (0.58) ACHEALDH1A1MAPK1MAPTHTT
SCHEMBL29543680 0.75 ACHE (0.58) ACHEALDH1A1MAPK1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2772480-B2 HIV REPLICATION INHIBITOR SHIONOGI & CO (JP) 2020-12-09 EP disclosed
EP-3204360-B1 THERAPEUTIC COMPOUNDS AND USES THEREOF GENENTECH INC (US) 2020-08-26 EP disclosed
EP-2772480-B1 HIV REPLICATION INHIBITOR SHIONOGI & CO (JP) 2018-05-23 EP disclosed
CN-1026206-C Arylpyrrole insecticidal acaricidal and nematicidal agents and method for preparation thereof AMERICAN CYANAMID CO (US) 1994-10-19 CN disclosed
CN-1039807-A Desinsection, kill mite, nematocides aryl-pyrrolidine and preparation method thereof AMERICAN CYANAMID CO (US) 1990-02-21 CN disclosed