SCHEMBL20171924

SCHEMBL20171924

CC(C)(C)Nc1nc(N2CCCC2)c2nc[nH]c2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.50
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
ALDH1A1 P00352 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
MAPK1 P28482 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
HTT P42858 4/20 0.37
TP53 P04637 1/20 0.37
ALOX15 P16050 1/20 0.36
AKT2 P31751 1/20 0.36
MAP3K5 Q99683 1/20 0.36
MAPT P10636 1/20 0.36
SLC29A1 Q99808 3/20 0.35
CNR2 P34972 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20171935 0.88 MAPK1 (0.43) LMNASMN1; SMN2NPSR1MAPK1HTT
SCHEMBL20171912 0.81 HTT (0.38) LMNAMEN1KMT2AALDH1A1CYP1A2
SCHEMBL16212037 0.81 CNR2 (0.56) CNR2
SCHEMBL16211714 0.79 CNR2 (0.54) CNR2
SCHEMBL2229901 0.79 NPY5R (0.43) LMNAMEN1KMT2AMAPK1L3MBTL1
SCHEMBL14071956 0.78 NPY5R (0.46) LMNAMEN1KMT2AMAPK1L3MBTL1
SCHEMBL20171876 0.76 HTT (0.41) LMNAALDH1A1SMN1; SMN2MAPK1HTT
SCHEMBL14183741 0.76 HTT (0.41) LMNAALDH1A1SMN1; SMN2MAPK1HTT
SCHEMBL8830247 0.76 CHUK (0.48) LMNAMAPK1HTTTP53ALOX15
SCHEMBL4513985 0.75 TLR7 (0.47) LMNAMEN1KMT2AALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2991987-B1 PURINE DERIVATIVES AS CB2 RECEPTOR AGONISTS HOFFMANN LA ROCHE (CH) 2018-05-23 EP disclosed