SCHEMBL20171959

SCHEMBL20171959

Cc1ncc(C#CCCCCl)c(Nc2ccccc2)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.38
EGFR P00533 2/20 0.38
BCL6 P41182 2/20 0.35
CYP3A4 P08684 3/20 0.34
MAPK1 P28482 1/20 0.34
JAK2 O60674 2/20 0.34
LRRK2 Q5S007 1/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C19 P33261 2/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
CYP2C9 P11712 1/20 0.34
APEX1 P27695 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CDK1 P06493 4/20 0.33
CDK2 P24941 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20171967 0.78 SYK (0.51) KDREGFRJAK2LRRK2CDK1
SCHEMBL6639897 0.72 EGFR (0.46) EGFRBCL6MAPK1JAK2LRRK2
SCHEMBL859187 0.70 EGFR (0.51) KDREGFRBCL6CYP3A4JAK2
SCHEMBL20171970 0.69 MERTK (0.51) KDREGFRJAK2CDK1CDK2
SCHEMBL30749051 0.66 MAP2K1 (0.59) KDRKDM4EMAPTCDK1AURKA
SCHEMBL5230508 0.65 EGFR (0.42) KDREGFRBCL6CYP3A4MAPK1
SCHEMBL20171963 0.65 SYK (0.49) KDRCYP1A2CYP2D6CYP2C19CYP2C9
SCHEMBL6644116 0.65 PIN1 (0.43) EGFRBCL6CDK1CDK2NPY5R
SCHEMBL6642666 0.65 PIN1 (0.51) KDREGFRBCL6MAPK1JAK2
SCHEMBL7714549 0.65 AURKA (0.41) KDREGFRBCL6CYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3323811-A1 PRODUCTION METHOD FOR NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, AND INTERMEDIATE OF SAID NITROGEN-CONTAINING HETEROCYCLIC COMPOUND FUJIFILM Corporation (JP) 2018-05-23 EP disclosed