SCHEMBL20172494

SCHEMBL20172494

FC(F)(F)c1ccc(Nc2cccnc2)nc1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.59
NPC1 O15118 3/20 0.56
RAB9A P51151 3/20 0.56
TDP1 Q9NUW8 1/20 0.56
IL1B P01584 1/20 0.50
NLRP3 Q96P20 1/20 0.50
CTSC P53634 1/20 0.47
TNNI3K Q59H18 1/20 0.46
EPHX2 P34913 1/20 0.46
KDM4E B2RXH2 1/20 0.45
GAA P10253 1/20 0.45
TRPV1 Q8NER1 1/20 0.45
CYP19A1 P11511 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17114620 0.83 NPC1 (0.63) NPC1RAB9ATNNI3KKDM4EGAA
SCHEMBL14577133 0.80 KIF11 (0.71) KIF11NPC1IL1BNLRP3CTSC
SCHEMBL20172492 0.80 KIF11 (0.66) KIF11IL1BNLRP3CTSC
SCHEMBL31013382 0.79 KIF11 (0.47) KIF11NPC1RAB9ATDP1IL1B
SCHEMBL31013379 0.78 KIF11 (0.46) KIF11NPC1RAB9ATDP1IL1B
SCHEMBL22970824 0.78 RAB9A (0.48) NPC1RAB9ATDP1GAATRPV1
SCHEMBL31013375 0.76 KIF11 (0.47) KIF11NPC1RAB9ATDP1IL1B
SCHEMBL22971132 0.76 KIF11 (0.60) KIF11IL1BNLRP3CTSCEPHX2
SCHEMBL10585521 0.76 KDM4E (0.55) NPC1RAB9ATDP1CTSCTNNI3K
SCHEMBL20172471 0.76 NPC1 (0.47) KIF11NPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3137459-B1 MORPHOLIN-PYRIDINE DERIVATIVES HAVING AFFINITY TO THE TAAR1 RECEPTOR HOFFMANN LA ROCHE (CH) 2018-05-23 EP disclosed