SCHEMBL20172492

SCHEMBL20172492

FC(F)(F)c1ccnc(Nc2cccnc2)c1

nearest known ligand 0.66

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.66
AURKA O14965 2/20 0.52
CTSC P53634 1/20 0.52
IL1B P01584 1/20 0.49
NLRP3 Q96P20 1/20 0.49
TSHR P16473 2/20 0.49
NOS3 P29474 1/20 0.49
NOS2 P35228 1/20 0.49
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
THRB P10828 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18672951 0.85 NPC1 (0.47) KIF11IL1BNLRP3KMT2AMEN1
SCHEMBL22971132 0.81 KIF11 (0.60) KIF11AURKACTSCIL1BNLRP3
SCHEMBL20172494 0.80 KIF11 (0.59) KIF11CTSCIL1BNLRP3
SCHEMBL22970832 0.80 ALOX15 (0.51) KIF11AURKATSHRNOS3NOS2
SCHEMBL4184375 0.78 AURKA (0.55) KIF11AURKACTSCNOS3NOS2
SCHEMBL31240789 0.76 ABL1 (0.48) KIF11CTSCKMT2AMEN1
SCHEMBL17969552 0.76 MAPK8 (0.45) KIF11TSHRKMT2AMEN1
SCHEMBL5748960 0.76 KARS1 (0.58) KIF11NOS2
SCHEMBL14577133 0.76 KIF11 (0.71) KIF11CTSCIL1BNLRP3TSHR
SCHEMBL1518621 0.75 MAPK10 (0.67) AURKAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3137459-B1 MORPHOLIN-PYRIDINE DERIVATIVES HAVING AFFINITY TO THE TAAR1 RECEPTOR HOFFMANN LA ROCHE (CH) 2018-05-23 EP disclosed