SCHEMBL2017353

SCHEMBL2017353

CCn1c(COC(=O)c2nc(Cl)c(N)nc2N)nc2cc(-c3ccc(OC)cc3)ccc21

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.52
NPC1 O15118 2/20 0.52
NLRP3 Q96P20 1/20 0.52
PPARG P37231 3/20 0.44
NPSR1 Q6W5P4 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C19 P33261 1/20 0.42
RAB9A P51151 1/20 0.42
TBXA2R P21731 2/20 0.40
NTRK1 P04629 2/20 0.40
CSF1R P07333 2/20 0.40
NTRK2 Q16620 2/20 0.40
SCNN1A P37088 4/20 0.39
TDP1 Q9NUW8 1/20 0.39
RPS6KA5 O75582 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2016915 0.94 MAPT (0.46) MAPTNPC1NLRP3PPARGNPSR1
SCHEMBL12635938 0.87 MAPT (0.46) MAPTNPC1NLRP3NPSR1CYP1A2
SCHEMBL2014103 0.86 SCNN1A (0.43) MAPTNPC1NLRP3PPARGSCNN1A
SCHEMBL12635760 0.82 SCNN1A (0.38) MAPTNPC1NLRP3PPARGSCNN1A
SCHEMBL2014866 0.81 SMN1; SMN2 (0.52) MAPTNPC1CYP1A2CYP3A4CYP2D6
Iodide SCHEMBL2016181 0.81 SCNN1A (0.38) MAPTNPC1NLRP3PPARGSCNN1A
SCHEMBL12636304 0.80 SCNN1A (0.38) MAPTNPC1NLRP3SCNN1A
Iodide SCHEMBL2018286 0.80 SCNN1A (0.38) MAPTNPC1NLRP3SCNN1A
SCHEMBL12635742 0.79 CHEK2 (0.41) MAPTNPC1NLRP3PPARGNPSR1
SCHEMBL2017964 0.79 SCNN1A (0.44) MAPTNPC1NLRP3PPARGCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed
WO-2011079087-A1 ENAC BLOCKERS GLAXO GROUP LIMITED (GB) 2011-06-30 WO disclosed