SCHEMBL20177137

SCHEMBL20177137

C=Cc1ccc(C(=C)c2cccc(C#N)c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.43
P4HB P07237 8/20 0.40
ENPP2 Q13822 1/20 0.38
GRIN2D O15399 2/20 0.37
GRIN3B O60391 2/20 0.37
GRIN1 Q05586 2/20 0.37
GRIN2A Q12879 2/20 0.37
GRIN2B Q13224 2/20 0.37
GRIN2C Q14957 2/20 0.37
GRIN3A Q8TCU5 2/20 0.37
ADORA2A P29274 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
FBP1 P09467 3/20 0.35
GRM5 P41594 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22359857 0.76 GSK3B (0.46) GSK3BENPP2GRIN2DGRIN3BGRIN1
SCHEMBL8383017 0.75 ALDH1A1 (0.56) ALDH1A1LMNAMAPT
SCHEMBL30601284 0.74 FBP1 (0.51) P4HBENPP2GRIN2DGRIN3BGRIN1
SCHEMBL471486 0.74 FBP1 (0.51) P4HBENPP2GRIN2DGRIN3BGRIN1
SCHEMBL10243324 0.73 CLK4 (0.47) CLK4
SCHEMBL16502093 0.72 GSK3B (0.53) GSK3BP4HBENPP2ADORA2ACLK4
Ethane SCHEMBL28057226 0.72 ALDH1A1 (0.52) ALDH1A1LMNAMAPT
SCHEMBL14508038 0.71 GSK3B (0.51) GSK3BP4HBENPP2CLK4FBP1
SCHEMBL3348656 0.71 GSK3B (0.51) GSK3BP4HBENPP2CLK4GRM5
SCHEMBL28080869 0.71 GSK3B (0.51) GSK3BP4HBENPP2CLK4GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093696-A1 INDAZOLE DERIVATIVES USEFUL AS INHIBITORS OF DIACYLGLYCERIDE O-ACYLTRANSFERASE 2 MERCK SHARP & DOHME CORP. (US) 2018-05-24 WO disclosed