SCHEMBL20177496

SCHEMBL20177496

Brc1ccc(C2Cc3nc4ccccc4n3C2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 3/20 0.44
MAPT P10636 2/20 0.44
BRD4 O60885 1/20 0.40
DPP4 P27487 1/20 0.37
DPP7 Q9UHL4 1/20 0.37
GALR3 O60755 1/20 0.37
NR2F2 P24468 1/20 0.37
ALDH1A1 P00352 1/20 0.37
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
TSHR P16473 2/20 0.36
POLB P06746 1/20 0.36
LMNA P02545 1/20 0.35
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 1/20 0.35
GFER P55789 1/20 0.35
KMT2A Q03164 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177639 1.00 GRM2 (0.44) GRM2MAPTBRD4DPP4DPP7
SCHEMBL20177500 0.79 DPP4 (0.43) GRM2MAPTDPP4DPP7ALDH1A1
SCHEMBL20177495 0.69 USP2 (0.40) GRM2MAPTGALR3NR2F2ALDH1A1
SCHEMBL20177558 0.68 GRM2 (0.45) GRM2MAPTDPP4DPP7ALDH1A1
SCHEMBL20177891 0.67 BRD4 (0.48) MAPTBRD4ALDH1A1ADRA1DADRA1A
SCHEMBL20177662 0.67 BRD4 (0.48) MAPTBRD4ALDH1A1ADRA1DADRA1A
SCHEMBL29941288 0.64 ALDH1A1 (0.40) GRM2DPP4DPP7ALDH1A1TSHR
SCHEMBL7924287 0.63 DPP4 (0.38) GRM2DPP4DPP7ALDH1A1MEN1
SCHEMBL5745617 0.62 TSHR (0.44) GRM2ALDH1A1TSHRNPC1RAB9A
SCHEMBL8355374 0.62 GRM2 (0.50) GRM2ALDH1A1TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed