SCHEMBL20177500

SCHEMBL20177500

Fc1cc(Br)cc(F)c1[C@H]1Cc2nc3ccccc3n2C1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 4/20 0.43
DPP7 Q9UHL4 1/20 0.43
GRM2 Q14416 8/20 0.36
MAPT P10636 1/20 0.36
CYP2D6 P10635 2/20 0.36
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34
KDM4E B2RXH2 1/20 0.34
TP53 P04637 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177558 0.84 GRM2 (0.45) DPP4DPP7GRM2MAPTALDH1A1
SCHEMBL20177639 0.79 GRM2 (0.44) DPP4DPP7GRM2MAPTALDH1A1
SCHEMBL20177496 0.79 GRM2 (0.44) DPP4DPP7GRM2MAPTALDH1A1
SCHEMBL20177640 0.72 DPP4 (0.38) DPP4DPP7ALDH1A1KDM4ETP53
SCHEMBL13342393 0.68 DPP4 (0.82) DPP4DPP7CYP2D6
SCHEMBL20177525 0.66 ADRA1A (0.56)
SCHEMBL20177859 0.66 ADRA1A (0.31)
SCHEMBL20177638 0.66 ADRA1A (0.56)
SCHEMBL7924287 0.62 DPP4 (0.38) DPP4DPP7GRM2ALDH1A1
SCHEMBL20177902 0.61 GRM4 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed