SCHEMBL20177522

SCHEMBL20177522

O=C1ONC2CC(c3ccc(Br)cc3)CN12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.41
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
NPC1 O15118 1/20 0.33
GAA P10253 1/20 0.33
MDM2 Q00987 1/20 0.32
KDM1A O60341 5/20 0.32
KCNH2 Q12809 2/20 0.32
MAOB P27338 2/20 0.32
RCOR1 Q9UKL0 2/20 0.32
KDM1B Q8NB78 1/20 0.32
ALDH1A1 P00352 3/20 0.32
HSD17B10 Q99714 1/20 0.31
LIG1 P18858 1/20 0.31
CHRNA7 P36544 2/20 0.31
TSHR P16473 1/20 0.31
CYP3A4 P08684 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177778 0.67 KDM4E (0.36) BRD4MEN1KMT2AGAAKDM1A
SCHEMBL28939724 0.61 BRD4 (0.43) BRD4MDM2ALDH1A1CHRNA7TSHR
SCHEMBL28939720 0.61 BRD4 (0.43) BRD4MDM2ALDH1A1CHRNA7TSHR
SCHEMBL5612 0.60 BRD4 (0.53) BRD4MEN1KMT2ANPC1GAA
SCHEMBL1673541 0.59 LMNA (0.49) BRD4CRBNMEN1KMT2ANPC1
SCHEMBL657720 0.59 BRD4 (0.49) BRD4MEN1KMT2ANPC1GAA
SCHEMBL5647940 0.59 BRD4 (0.44) BRD4GAAKDM1AKCNH2MAOB
SCHEMBL23119770 0.58 BRD4 (0.47) BRD4KDM1AKCNH2MAOBRCOR1
SCHEMBL20341692 0.58 BRD4 (0.47) BRD4MEN1KMT2ANPC1GAA
SCHEMBL265495 0.58 KDM1A (0.48) BRD4KDM1AKCNH2MAOBRCOR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed