SCHEMBL28939720

SCHEMBL28939720

CN1C(=O)C2CC(c3ccc(Br)cc3)CN2c2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.43
EGFR P00533 1/20 0.37
CHRNA7 P36544 2/20 0.36
CYP3A4 P08684 3/20 0.35
CYP2C9 P11712 3/20 0.35
CYP2C19 P33261 2/20 0.35
TSHR P16473 2/20 0.35
LMNA P02545 1/20 0.35
ALOX15 P16050 1/20 0.35
MAPK1 P28482 1/20 0.35
CCKBR P32239 4/20 0.35
CCKAR P32238 3/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28939724 1.00 BRD4 (0.43) BRD4EGFRCHRNA7CYP3A4CYP2C9
SCHEMBL28940152 0.85 MAPT (0.36) BRD4EGFRALOX15ALDH1A1
SCHEMBL28940153 0.85 MAPT (0.36) BRD4EGFRALOX15ALDH1A1
SCHEMBL20177778 0.66 KDM4E (0.36) BRD4CYP3A4CYP2C9CYP2C19TSHR
SCHEMBL28940083 0.64 ALDH1A1 (0.37) EGFRTSHRMAPK1CCKBRGABRP
SCHEMBL30095518 0.63 GABRA1 (0.39) BRD4CYP3A4CYP2C9CYP2C19TSHR
SCHEMBL28940149 0.63 GABRA1 (0.39) BRD4CYP3A4CYP2C9CYP2C19TSHR
Hydrochloric Acid SCHEMBL6421986 0.61 HTR2C (0.49) CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL20177522 0.61 BRD4 (0.41) BRD4CHRNA7CYP3A4CYP2C9CYP2C19
SCHEMBL20177851 0.60 BRD4 (0.54) BRD4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115637454-A Synthesis method of tetrahydroimidazo [1,5-a ] quinoxaline-4 (5H) -one derivative 南华大学 2023-01-24 CN disclosed