SCHEMBL20177778

SCHEMBL20177778

Brc1ccc([C@H]2CC3Nc4ccccc4N3C2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.36
MAPT P10636 3/20 0.36
ALDH1A1 P00352 3/20 0.36
LMNA P02545 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
RECQL P46063 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
HTT P42858 2/20 0.36
POLB P06746 1/20 0.36
XBP1 P17861 1/20 0.36
BRD4 O60885 2/20 0.34
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2D6 P10635 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177564 0.79 KDM1A (0.32) KDM1A
SCHEMBL20177515 0.68 SMN1; SMN2 (0.35) ALDH1A1SMN1; SMN2BRD4MAPK1MEN1
SCHEMBL20177522 0.67 BRD4 (0.41) MAPTALDH1A1BRD4CYP3A4CYP2C9
Acetic Acid SCHEMBL6476155 0.66 GAA (0.43) KDM4EMAPTALDH1A1SMN1; SMN2TDP1
SCHEMBL28939720 0.66 BRD4 (0.43) ALDH1A1LMNABRD4CYP3A4CYP2C9
SCHEMBL28939724 0.66 BRD4 (0.43) ALDH1A1LMNABRD4CYP3A4CYP2C9
SCHEMBL29616904 0.65 BRD4 (0.41) KDM4EMAPTALDH1A1LMNASMN1; SMN2
SCHEMBL28736993 0.65 BRD4 (0.41) KDM4EMAPTALDH1A1LMNASMN1; SMN2
SCHEMBL28736992 0.65 BRD4 (0.41) KDM4EMAPTALDH1A1LMNASMN1; SMN2
SCHEMBL457928 0.63 RAB9A (0.49) KDM4EMAPTALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed