SCHEMBL20177536

SCHEMBL20177536

N[C@@H]1C2=NOCCN2C[C@H]1c1ccc(Br)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 7/20 0.40
MAOB P27338 4/20 0.40
KCNH2 Q12809 2/20 0.40
RCOR1 Q9UKL0 2/20 0.40
KDM1B Q8NB78 1/20 0.40
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
PKM P14618 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
THPO P40225 1/20 0.33
MAPK1 P28482 2/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177590 0.86 CYP1A2 (0.33) KDM1AMAOBHTR2CHTR2BCYP1A2
SCHEMBL20177889 0.80 KDM1A (0.48) KDM1AKDM1BFPR2
SCHEMBL20177610 0.69 BRD4 (0.41) CYP1A2CYP3A4PKMTSHRNFKB1
SCHEMBL20177535 0.69 BRD4 (0.41) CYP1A2CYP3A4PKMTSHRNFKB1
SCHEMBL20177614 0.68 CTSL (0.42) KDM1AMAOBRCOR1KDM1BTSHR
SCHEMBL20177495 0.60 USP2 (0.40) KDM1AMAOBKCNH2RCOR1KDM1B
SCHEMBL5454146 0.60 KDM1A (0.50) KDM1AMAOBKCNH2RCOR1KDM1B
SCHEMBL5454149 0.60 KDM1A (0.50) KDM1AMAOBKCNH2RCOR1KDM1B
SCHEMBL5454142 0.60 KDM1A (0.50) KDM1AMAOBKCNH2RCOR1KDM1B
SCHEMBL16019172 0.60 KDM1A (1.00) KDM1AMAOBKCNH2RCOR1KDM1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed