SCHEMBL20177569

SCHEMBL20177569

O/N=C1/CC(c2ccc(Br)cc2)CN1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.37
BRD4 O60885 1/20 0.36
TSHR P16473 2/20 0.33
KDM1A O60341 5/20 0.32
KCNH2 Q12809 2/20 0.32
MAOB P27338 2/20 0.32
RCOR1 Q9UKL0 2/20 0.32
KDM1B Q8NB78 1/20 0.32
MAPT P10636 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ESRRG P62508 1/20 0.32
LMNA P02545 1/20 0.31
MAP1LC3B Q9GZQ8 1/20 0.31
PKM P14618 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177592 0.76 ESRRG (0.34) ESR2BRD4TSHRESRRG
SCHEMBL20177606 0.73 TSHR (0.57) BRD4TSHRPKMGAA
SCHEMBL481990 0.73 TSHR (0.57) BRD4TSHRPKMGAA
SCHEMBL11080147 0.69 GABRP (0.39) BRD4KDM1AKCNH2MAOBRCOR1
SCHEMBL12540718 0.67 ESR2 (0.56) ESR2BRD4KDM1AKCNH2MAOB
SCHEMBL12540716 0.67 ESR2 (0.56) ESR2BRD4KDM1AKCNH2MAOB
SCHEMBL12540720 0.67 ESR2 (0.56) ESR2BRD4KDM1AKCNH2MAOB
SCHEMBL15301182 0.66 ESRRG (0.48) BRD4KDM1AKCNH2MAOBRCOR1
SCHEMBL12814549 0.66 MAP1LC3B (0.44) BRD4MAPTSMN1; SMN2LMNAMAP1LC3B
SCHEMBL12382040 0.66 BRD4 (0.33) BRD4KDM1AKCNH2MAOBRCOR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed