SCHEMBL20177592

SCHEMBL20177592

OCCO/N=C1/C[C@H](c2ccc(Br)cc2)CN1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESRRG P62508 1/20 0.34
ESR2 Q92731 1/20 0.31
TSHR P16473 1/20 0.30
GPBAR1 Q8TDU6 1/20 0.30
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177943 0.86 HTR3A (0.36) ESR2TSHRGPBAR1
SCHEMBL16785342 0.84 TSHR (0.40) TSHR
SCHEMBL19559484 0.84 TSHR (0.40) TSHR
SCHEMBL20177882 0.80 KDM1A (0.35)
SCHEMBL20177855 0.78
SCHEMBL20177569 0.76 ESR2 (0.37) ESRRGESR2TSHRBRD4
SCHEMBL20177534 0.76 RECQL (0.31) GPBAR1
SCHEMBL20177801 0.75 ALDH1A1 (0.34) ESR2
SCHEMBL20177903 0.70
SCHEMBL20041973 0.70 TSHR (0.39) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed