SCHEMBL20177579

SCHEMBL20177579

O=C1C[C@H](c2cc(F)c(Cl)cc2F)CN1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.44
KDM1B Q8NB78 1/20 0.44
MTNR1A P48039 2/20 0.42
SCN8A Q9UQD0 2/20 0.38
IDO1 P14902 2/20 0.38
PDE4A P27815 3/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
TSHR P16473 1/20 0.37
FPR1 P21462 4/20 0.36
FPR2 P25090 3/20 0.36
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29869025 0.86 MTNR1A (0.46) MTNR1APDE4AALDH1A1CYP1A2CYP2C19
SCHEMBL18590496 0.81 MTNR1A (0.42) MTNR1AIDO1PDE4AALDH1A1CYP1A2
SCHEMBL20177679 0.81 KDM1A (0.44) KDM1AKDM1BIDO1ALDH1A1HTR2A
SCHEMBL20177704 0.79 MTNR1A (0.48) MTNR1ASCN8APDE4AALDH1A1CYP1A2
SCHEMBL19559449 0.77 PDE4A (0.54) MTNR1APDE4AALDH1A1CYP1A2PDE4B
SCHEMBL19559393 0.77 PDE4A (0.54) MTNR1APDE4AALDH1A1CYP1A2PDE4B
SCHEMBL19559446 0.76 LMNA (0.43) MTNR1APDE4AALDH1A1CYP1A2CYP2C19
SCHEMBL16785506 0.76 LMNA (0.43) MTNR1APDE4AALDH1A1CYP1A2CYP2C19
SCHEMBL12498577 0.76 PDE4A (0.52) PDE4AALDH1A1CYP1A2CYP2C19PDE4B
SCHEMBL12498580 0.76 PDE4A (0.52) PDE4AALDH1A1CYP1A2CYP2C19PDE4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed