SCHEMBL20177704

SCHEMBL20177704

O=C1C[C@H](c2ccc(Cl)cc2F)CN1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.48
FPR1 P21462 4/20 0.45
FPR2 P25090 3/20 0.45
GPBAR1 Q8TDU6 1/20 0.41
SCN8A Q9UQD0 2/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
OPRL1 P41146 3/20 0.39
PDE4A P27815 3/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
TSHR P16473 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
PROKR1 Q8TCW9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15549178 0.84 MTNR1A (0.50) MTNR1AFPR1FPR2HTR2AHTR2C
SCHEMBL20177918 0.81 HTR2C (0.40) FPR1FPR2GPBAR1HTR2AHTR2C
SCHEMBL560175 0.81 MTNR1A (0.48) MTNR1AFPR1FPR2HTR2CPDE4A
SCHEMBL18590494 0.81 MTNR1A (0.48) MTNR1APDE4AALDH1A1CYP1A2CYP2C19
SCHEMBL559712 0.81 MTNR1A (0.48) MTNR1AFPR1FPR2HTR2CPDE4A
SCHEMBL559629 0.81 MTNR1A (0.48) MTNR1AFPR1FPR2HTR2CPDE4A
SCHEMBL20177600 0.81 MTNR1A (0.48) MTNR1AFPR1FPR2PDE4AALDH1A1
Hydrochloric Acid SCHEMBL560453 0.80 MTNR1A (0.47) MTNR1AFPR1FPR2HTR2CPDE4A
SCHEMBL20177579 0.79 KDM1A (0.44) MTNR1AFPR1FPR2SCN8AHTR2A
SCHEMBL560148 0.79 MTNR1A (0.46) MTNR1AFPR1FPR2HTR2CPDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed