SCHEMBL20177582

SCHEMBL20177582

COC1=NCC(c2c(F)cc(OC)cc2F)C1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.39
KDM1A O60341 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
FPR2 P25090 9/20 0.32
FPR1 P21462 5/20 0.32
CPS1 P31327 5/20 0.32
ALDH1A1 P00352 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
CYP1A1 P04798 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP1B1 Q16678 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177908 0.86
SCHEMBL19559545 0.80 FPR2 (0.33) TAAR1KDM1AMAOAMAOBFPR2
SCHEMBL19559483 0.74 FPR1 (0.40) KDM1AMAOAMAOBFPR2FPR1
SCHEMBL20177609 0.73 FPR2 (0.31) TAAR1FPR2
SCHEMBL20041817 0.70 GCK (0.35) FPR2FPR1
SCHEMBL18117745 0.70 GCK (0.35) FPR2FPR1
SCHEMBL16785337 0.67 PDE4A (0.49) FPR2FPR1
SCHEMBL20177630 0.67 FPR1 (0.38) TAAR1FPR2FPR1
SCHEMBL19559455 0.67 PDE4A (0.49) FPR2FPR1
SCHEMBL19559459 0.66 PDE4A (0.50) FPR1CPS1ALDH1A1HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed