SCHEMBL20177653

SCHEMBL20177653

O=C1C[C@H](c2ccc(Br)cc2)CN1c1ccccc1[N+](=O)[O-]

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 7/20 0.48
BRD4 O60885 5/20 0.48
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.41
HTT P42858 2/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
HSP90AB1 P08238 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177848 0.81 ALDH1A1 (0.39) GSK3BALDH1A1MAPTHTTLMNA
SCHEMBL20177851 0.80 BRD4 (0.54) BRD4MAPTPDE4APDE4BPDE4C
SCHEMBL20177560 0.71 ALDH1A1 (0.43) ALDH1A1MAPTLMNAKMT2APDE4A
SCHEMBL11183526 0.68 ALDH1A1 (0.50) GSK3BALDH1A1MAPTHTTLMNA
SCHEMBL23043784 0.66 HTT (0.54) ALDH1A1MAPTHTTLMNAKMT2A
SCHEMBL29740649 0.65 MAPT (0.47) ALDH1A1MAPTHTTLMNAKMT2A
SCHEMBL1628707 0.65 MAPT (0.47) ALDH1A1MAPTHTTLMNAKMT2A
SCHEMBL10620885 0.65 MAPT (0.53) GSK3BALDH1A1MAPTHTTLMNA
SCHEMBL29978521 0.65 HTT (0.52) GSK3BALDH1A1MAPTHTTLMNA
SCHEMBL23043626 0.65 HTT (0.52) GSK3BALDH1A1MAPTHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed