SCHEMBL20177560

SCHEMBL20177560

COc1cc(F)c(C2CC(=O)N(c3ccccc3[N+](=O)[O-])C2)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
MAPT P10636 4/20 0.40
GAA P10253 1/20 0.39
ACHE P22303 1/20 0.38
BACE1 P56817 1/20 0.38
GFER P55789 1/20 0.38
TP53 P04637 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
CYP19A1 P11511 1/20 0.37
GRM5 P41594 1/20 0.37
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177848 0.86 ALDH1A1 (0.39) ALDH1A1KMT2AMAPTSMN1; SMN2GRM5
SCHEMBL20177834 0.83 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL24184779 0.72 GRM5 (0.36) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL20177653 0.71 GSK3B (0.48) ALDH1A1KMT2APDE4APDE4BPDE4C
SCHEMBL18117769 0.71 PDE4A (0.50) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL19559459 0.71 PDE4A (0.50) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL24257180 0.70 POLB (0.33) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL24184129 0.70 PDE4A (0.35) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL24257179 0.70 POLB (0.33) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL19559422 0.70 HCRTR1 (0.38) PDE4APDE4BPDE4CPDE4DMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed