SCHEMBL20177899

SCHEMBL20177899

COc1ccc(COC(=O)N[C@@H]2C(=O)N(c3ccccc3N)C[C@H]2c2c(F)cc(Br)cc2F)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 8/20 0.40
KCNQ2 O43526 1/20 0.38
PKM P14618 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TSHR P16473 1/20 0.37
FPR1 P21462 2/20 0.37
FPR2 P25090 2/20 0.37
CYP2D6 P10635 2/20 0.36
MAPT P10636 2/20 0.36
ATM Q13315 1/20 0.36
P2RX4 Q99571 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
ACHE P22303 1/20 0.35
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
BRD3 Q15059 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177832 0.90 CA1 (0.43) CYP3A4KCNQ2TSHRFPR1FPR2
SCHEMBL20177846 0.87 KDM1A (0.40) CYP3A4KCNQ2PKMHTTSMN1; SMN2
SCHEMBL20177594 0.77 FPR2 (0.59) CYP3A4FPR1FPR2
SCHEMBL20177499 0.76 SMN1; SMN2 (0.37) KCNQ2PKMHTTSMN1; SMN2MAPT
SCHEMBL18106745 0.75 CA1 (0.47) KCNQ2FPR1FPR2CA1CA2
SCHEMBL18106743 0.75 CA1 (0.47) KCNQ2FPR1FPR2CA1CA2
SCHEMBL29434434 0.75 CA1 (0.47) KCNQ2FPR1FPR2CA1CA2
SCHEMBL20177604 0.75 FPR2 (0.47) CYP3A4KCNQ2PKMHTTSMN1; SMN2
SCHEMBL16785496 0.74 FPR1 (0.47) CYP3A4KCNQ2TSHRFPR1FPR2
SCHEMBL29434315 0.74 FPR1 (0.47) CYP3A4KCNQ2TSHRFPR1FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed