SCHEMBL20177499

SCHEMBL20177499

COc1ccc(COC(=O)N[C@@H]2c3nc4ccccc4n3C[C@H]2c2c(F)cc(Br)cc2F)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.37
PKM P14618 1/20 0.37
HTT P42858 1/20 0.37
GSK3B P49841 1/20 0.37
NPC1 O15118 1/20 0.37
KDM4E B2RXH2 1/20 0.37
CNR2 P34972 3/20 0.36
MAPT P10636 2/20 0.36
KCNQ2 O43526 1/20 0.36
GAA P10253 2/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.35
ATM Q13315 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
ACHE P22303 1/20 0.35
KCNH2 Q12809 1/20 0.35
TACR2 P21452 1/20 0.35
TACR1 P25103 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20177557 0.90 CA1 (0.42) NPC1KCNQ2CA1CA2ACHE
SCHEMBL20177642 0.88 SMN1; SMN2 (0.39) SMN1; SMN2PKMHTTGSK3BNPC1
SCHEMBL20177613 0.76 FPR2 (0.58) SMN1; SMN2PKMHTTMAPTALDH1A1
SCHEMBL20177899 0.76 CYP3A4 (0.40) SMN1; SMN2PKMHTTMAPTKCNQ2
SCHEMBL20177594 0.75 FPR2 (0.59)
SCHEMBL20177845 0.75 BRD4 (0.47) NPC1KCNQ2CA1CA2ACHE
SCHEMBL20177563 0.74 FPR2 (0.45) HTTNPC1MAPTGAAALDH1A1
SCHEMBL20177604 0.74 FPR2 (0.47) SMN1; SMN2PKMHTTKCNQ2ALDH1A1
SCHEMBL20177512 0.74 FPR2 (0.59)
SCHEMBL20177909 0.73 BRD4 (0.43) NPC1KCNQ2CA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018092916-A1 NITROGEN-CONTAINING POLYCYCLIC HETEROCYCLIC DERIVATIVE 宇部興産株式会社 2018-05-24 WO disclosed