SCHEMBL20179460

SCHEMBL20179460

CCN(C(=O)CCCCCNS(C)(=O)=O)[C@@H](C)C(=O)NCc1cccs1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP2 O75604 1/20 0.43
GAA P10253 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
ALDH1A1 P00352 3/20 0.39
TSHR P16473 3/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PKM P14618 1/20 0.38
F12 P00748 3/20 0.38
POLB P06746 1/20 0.37
HTT P42858 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20179555 0.75 HPGD (0.62) GAANPSR1ALDH1A1TSHRMEN1
SCHEMBL20179556 0.71 CTSK (0.48) GAANPSR1CYP3A4CYP2D6CYP2C19
SCHEMBL20179646 0.71 GAA (0.43) GAANPSR1ALDH1A1TSHRMEN1
SCHEMBL20179732 0.69 USP2 (0.45) USP2GAANPSR1ALDH1A1TSHR
SCHEMBL1107021 0.67 GAA (0.62) USP2GAANPSR1ALDH1A1TSHR
SCHEMBL28820376 0.66 USP2 (0.67) USP2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL24799334 0.66 USP2 (0.44) USP2GAANPSR1ALDH1A1TSHR
SCHEMBL10253878 0.66 GAA (0.60) USP2GAANPSR1ALDH1A1TSHR
SCHEMBL17397492 0.66 POLB (0.41) USP2GAANPSR1ALDH1A1TSHR
SCHEMBL5298689 0.65 KMT2A (0.59) GAAALDH1A1TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093695-A1 FACTOR XIIa INHIBITORS MERCK SHARP & DOHME CORP. (US) 2018-05-24 WO disclosed