SCHEMBL20179555

SCHEMBL20179555

CCN(C(=O)CCC1CCCCC1)[C@@H](C)C(=O)NCc1cccs1

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.62
KMT2A Q03164 3/20 0.60
MEN1 O00255 2/20 0.60
CTSK P43235 1/20 0.46
GPR88 Q9GZN0 1/20 0.44
GAA P10253 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
POLB P06746 1/20 0.44
ALDH1A1 P00352 5/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
TSHR P16473 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ADAM17 P78536 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20179646 0.81 GAA (0.43) HPGDKMT2AMEN1CTSKGPR88
SCHEMBL6076593 0.78 HPGD (1.00) HPGDKMT2AMEN1POLBALDH1A1
SCHEMBL20179645 0.76 GPR88 (0.41) HPGDKMT2AMEN1CTSKGPR88
SCHEMBL6075693 0.76 KMT2A (1.00) HPGDKMT2AMEN1POLBALDH1A1
SCHEMBL20179556 0.75 CTSK (0.48) HPGDKMT2AMEN1CTSKGAA
SCHEMBL20179460 0.75 USP2 (0.43) KMT2AMEN1GAANPSR1POLB
SCHEMBL7355924 0.70 METAP2 (0.60) HPGDKMT2AMEN1CTSKPOLB
SCHEMBL1107021 0.69 GAA (0.62) HPGDKMT2AMEN1GAANPSR1
Hydrochloric Acid SCHEMBL7355919 0.69 METAP2 (0.59) HPGDKMT2AMEN1CTSKPOLB
SCHEMBL24799563 0.69 HPGD (0.58) HPGDKMT2AMEN1GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093695-A1 FACTOR XIIa INHIBITORS MERCK SHARP & DOHME CORP. (US) 2018-05-24 WO disclosed