SCHEMBL20179696

SCHEMBL20179696

CN1CCC(Oc2ccc(C(=O)C(Br)c3ccc(OCc4ccccc4)cc3)cc2)C1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.55
ACACB O00763 3/20 0.54
CHRM4 P08173 1/20 0.47
CHRNB2 P17787 1/20 0.46
CHRNA5 P30532 1/20 0.46
CHRNA7 P36544 1/20 0.46
CHRNA4 P43681 1/20 0.46
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
SLC6A5 Q9Y345 1/20 0.44
KDM4E B2RXH2 2/20 0.44
MAOB P27338 1/20 0.44
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
CCR5 P51681 1/20 0.43
EGFR P00533 2/20 0.43
MEN1 O00255 1/20 0.43
MAPK1 P28482 1/20 0.43
KMT2A Q03164 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20165040 0.86 ESR1 (0.48) MCHR1ACACBKDM4EALDH1A1LMNA
SCHEMBL20179666 0.86 ESR1 (0.48) MCHR1ACACBKDM4EALDH1A1LMNA
SCHEMBL20165043 0.86 ESR1 (0.48) MCHR1ACACBKDM4EALDH1A1LMNA
SCHEMBL20179695 0.82 MCHR1 (0.58) MCHR1ACACBCHRNB2CHRNA5CHRNA7
SCHEMBL13772738 0.79 NR4A1 (0.62) MAOBALDH1A1LMNAEGFRNR4A1
SCHEMBL6210392 0.79 RAB9A (0.58) MAOBALDH1A1NR4A1NR4A2NR4A3
SCHEMBL6208904 0.79 RAB9A (0.58) MAOBALDH1A1NR4A1NR4A2NR4A3
SCHEMBL3270043 0.74 NR4A1 (0.55) MAOBALDH1A1LMNAEGFRNR4A1
SCHEMBL26815710 0.73 RXRB (0.53) SLC6A5MAOBNR4A1NR4A2NR4A3
SCHEMBL14487845 0.72 CHRNB2 (0.54) CHRNB2CHRNA5CHRNA7CHRNA4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018091153-A1 NOVEL SUBSTITUTED N-(3-FLUOROPROPYL)-PYRROLIDINE COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND THERAPEUTIC USES THEREOF SANOFI (FR) 2018-05-24 WO disclosed