SCHEMBL20180161

SCHEMBL20180161

N=Cc1cc(-c2ccncc2)ccc1Nc1cccc(Br)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 2/20 0.43
PTGS2 P35354 2/20 0.43
EGFR P00533 6/20 0.41
PKMYT1 Q99640 1/20 0.41
ALK Q9UM73 1/20 0.40
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
PKM P14618 1/20 0.39
KMT2A Q03164 1/20 0.39
BUB1 O43683 1/20 0.37
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
GAK O14976 1/20 0.37
FLT1 P17948 1/20 0.36
KDR P35968 1/20 0.36
GRK2 P25098 1/20 0.35
ERN1 O75460 1/20 0.35
RAPGEF4 Q8WZA2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20180167 0.88 NPC1 (0.38) PTGS1PTGS2EGFRALKMEN1
SCHEMBL20180309 0.88 ABCG2 (0.41) EGFRALKMEN1KMT2AKDR
SCHEMBL20180229 0.81 MEN1 (0.40) EGFRALKMEN1NPC1KMT2A
SCHEMBL20180158 0.79 EGFR (0.38) EGFRPKMYT1ALKBUB1KDR
SCHEMBL20180549 0.76 EGFR (0.47) PTGS1PTGS2EGFRMEN1KMT2A
SCHEMBL20180257 0.72 FBP1 (0.44) PTGS1PTGS2EGFRMEN1KMT2A
SCHEMBL20180162 0.72 ACP1 (0.42) ALKMEN1KMT2AKDR
SCHEMBL22927246 0.72 BRAF (0.50) PKMYT1MEN1KMT2A
SCHEMBL20180153 0.72 ALK (0.41) PTGS1PTGS2EGFRPKMYT1ALK
SCHEMBL19624969 0.71 ALK (0.45) PTGS1PTGS2ALKMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018093107-A1 ORGANIC COMPOUND AND ORGANIC ELECTROLUMINESCENT ELEMENT COMPRISING SAME 주식회사 두산 2018-05-24 WO disclosed