SCHEMBL20180554

SCHEMBL20180554

CN1CCN(c2c(Cl)cc(I)cc2Cl)CC1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.47
MAPT P10636 1/20 0.47
RAD52 P43351 1/20 0.47
DRD2 P14416 2/20 0.42
DRD3 P35462 2/20 0.42
HRH4 Q9H3N8 5/20 0.41
POLB P06746 1/20 0.40
BCL2A1 Q16548 1/20 0.38
HTR1A P08908 1/20 0.37
DRD4 P21917 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
HTR3E A5X5Y0 2/20 0.37
HTR3B O95264 2/20 0.37
HTR3A P46098 2/20 0.37
HTR3D Q70Z44 2/20 0.37
HTR3C Q8WXA8 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20180543 0.85 SMN1; SMN2 (0.42) KDM4EMAPTRAD52DRD2DRD3
SCHEMBL21388466 0.82 HRH4 (0.46) KDM4EMAPTRAD52DRD2DRD3
SCHEMBL10126855 0.80 KDM4E (0.61) KDM4EMAPTRAD52DRD2DRD3
SCHEMBL13416764 0.80 CCR4 (0.43) KDM4EMAPTRAD52DRD2DRD3
SCHEMBL20180555 0.78 KDM4E (0.64) KDM4EMAPTRAD52DRD2DRD3
SCHEMBL20180762 0.78 MAPT (0.39) KDM4EMAPTRAD52HRH4POLB
SCHEMBL25675632 0.77 HRH4 (0.45) KDM4EMAPTRAD52DRD2DRD3
SCHEMBL13416761 0.77 HRH4 (0.46) KDM4EMAPTRAD52DRD2DRD3
SCHEMBL17340291 0.76 SMN1; SMN2 (0.42) KDM4EMAPTRAD52DRD2DRD3
SCHEMBL17690602 0.76 MAPT (0.40) KDM4EMAPTRAD52DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018090939-A1 8,9-DIHYDROIMIDAZOLE[1,2-A]PYRIMIDO[5,4-E]PYRIMIDINE-5(6H)-KETONE COMPOUND 上海瑛派药业有限公司 2018-05-24 WO disclosed