SCHEMBL17690602

SCHEMBL17690602

CN1CCN(c2c(Cl)cc(N=O)cc2Cl)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
RAD52 P43351 1/20 0.40
HRH4 Q9H3N8 3/20 0.39
DRD2 P14416 3/20 0.39
DRD3 P35462 3/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
NPC1 O15118 1/20 0.37
THRB P10828 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 1/20 0.37
BCL2A1 Q16548 3/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
BCL2 P10415 1/20 0.36
ALOX12 P18054 1/20 0.36
BID P55957 1/20 0.36
RAD51 Q06609 1/20 0.36
BCL2L1 Q07817 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21388466 0.77 HRH4 (0.46) MAPTKDM4ERAD52HRH4DRD2
SCHEMBL20180554 0.76 KDM4E (0.47) MAPTKDM4ERAD52HRH4DRD2
SCHEMBL13416764 0.76 CCR4 (0.43) MAPTKDM4ERAD52HRH4DRD2
SCHEMBL10126855 0.76 KDM4E (0.61) MAPTKDM4ERAD52HRH4DRD2
SCHEMBL13416761 0.73 HRH4 (0.46) MAPTKDM4ERAD52HRH4DRD2
SCHEMBL25675632 0.73 HRH4 (0.45) MAPTKDM4ERAD52HRH4DRD2
SCHEMBL10126859 0.72 SIRT6 (0.54) MAPTL3MBTL1SMN1; SMN2POLBBCL2A1
SCHEMBL17340291 0.71 SMN1; SMN2 (0.42) MAPTKDM4ERAD52HRH4DRD2
SCHEMBL21448015 0.71 DRD2 (0.63) MAPTKDM4ERAD52HRH4DRD2
SCHEMBL1938752 0.69 ADRB2 (0.60) MAPTKDM4ERAD52HRH4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3009428-A1 DIAMINO HETEROCYCLIC CARBOXAMIDE COMPOUND Astellas Pharma Inc. (JP) 2016-04-20 EP disclosed