SCHEMBL20182191

SCHEMBL20182191

CCC(/C(=C/Nc1ccc(F)cc1)N=N)n1cc(-c2cncnc2OC)c2c(N)ncnc21

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.34
CFTR P13569 3/20 0.33
AXL P30530 5/20 0.33
EGFR P00533 3/20 0.33
MET P08581 4/20 0.32
KDR P35968 2/20 0.32
TEK Q02763 2/20 0.32
ABL1 P00519 2/20 0.32
ABL2 P42684 2/20 0.32
RET P07949 1/20 0.32
EIF2AK3 Q9NZJ5 1/20 0.31
SRC P12931 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182271 0.93 CFTR (0.35) ALKCFTRAXLEGFRKDR
SCHEMBL20182224 0.92 EGFR (0.39) CFTREGFRKDRTEKABL1
SCHEMBL20182265 0.90 NTRK1 (0.36) ALKCFTRAXLEGFRKDR
SCHEMBL20181916 0.89 CFTR (0.39) CFTREGFRKDRTEKABL1
SCHEMBL20182222 0.85 AXL (0.34) AXLEGFRKDRTEKABL1
SCHEMBL20182226 0.84 BTK (0.35) CFTREGFRABL1ABL2EIF2AK3
SCHEMBL20182275 0.82 EGFR (0.36) AXLEGFRKDRTEKABL1
SCHEMBL20182235 0.82 EIF2AK3 (0.34) AXLEGFRKDRTEKABL1
SCHEMBL20182289 0.82 NTRK1 (0.36) AXLEGFRKDRTEKABL1
SCHEMBL20182175 0.82 DYRK3 (0.35) AXLMETRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed