SCHEMBL20182175

SCHEMBL20182175

CCC(/C(=C/Nc1ccc(F)cc1)N=N)n1cc(I)c2c(N)ncnc21

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK3 O43781 1/20 0.35
ROCK2 O75116 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35
PHKG2 P15735 1/20 0.35
PRKACA P17612 1/20 0.35
RPS6KB1 P23443 1/20 0.35
MARK3 P27448 1/20 0.35
FLT3 P36888 1/20 0.35
CSNK1A1 P48729 1/20 0.35
CSNK1D P48730 1/20 0.35
CLK2 P49760 1/20 0.35
IRAK1 P51617 1/20 0.35
CSNK1G2 P78368 1/20 0.35
MAP4K2 Q12851 1/20 0.35
ROCK1 Q13464 1/20 0.35
CAMK2G Q13555 1/20 0.35
CAMK2D Q13557 1/20 0.35
DYRK1A Q13627 1/20 0.35
MELK Q14680 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182191 0.82 ALK (0.34) METAXLRET
SCHEMBL20182248 0.77 LRRK2 (0.34) ROCK2MAP4K4RPS6KB1FLT3CLK2
SCHEMBL20182296 0.76 CFTR (0.41)
SCHEMBL20182225 0.76 CFTR (0.39) FLT3AXLRET
SCHEMBL20182291 0.76 NTRK1 (0.38) FLT3METAXLNTRK1NTRK3
SCHEMBL20182222 0.76 AXL (0.34) FLT3AXLRET
SCHEMBL20182275 0.75 EGFR (0.36) FLT3AXLRET
SCHEMBL20182271 0.74 CFTR (0.35) AXLRET
SCHEMBL20182292 0.74 NEK7 (0.37) FLT3NTRK1NTRK3NTRK2
SCHEMBL20182234 0.74 EGFR (0.35) FLT3RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018094137-A1 PYRROLOPYRIMIDINES AS CFTR POTENTIATORS CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC. (US) 2018-05-24 WO disclosed