SCHEMBL20182714

SCHEMBL20182714

CCS(=O)(=O)c1cc(-c2cccc(F)c2)cnc1-c1nc2cc(C(F)(F)F)cnc2n1C

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.40
GRIN1 Q05586 16/20 0.40
GRIN2B Q13224 16/20 0.40
PTGS2 P35354 2/20 0.40
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
PTGS1 P23219 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20182758 0.92 POLB (0.44) POLBGRIN1GRIN2BPTGS2USP2
SCHEMBL20182759 0.89 POLB (0.43) POLBGRIN1GRIN2BPTGS2
SCHEMBL21641516 0.86 POLB (0.45) POLBUSP2ALDH1A1CYP1A2CLK4
SCHEMBL14684583 0.86 POLB (0.48) POLBALDH1A1
SCHEMBL29360277 0.86 POLB (0.48) POLBALDH1A1
SCHEMBL18866344 0.86 POLB (0.42) POLBGRIN1GRIN2BPTGS2ALDH1A1
SCHEMBL15868301 0.83 POLB (0.46) POLBALDH1A1
SCHEMBL25885629 0.83 POLB (0.39) POLBGRIN1GRIN2B
SCHEMBL30989728 0.83 POLB (0.39) POLBGRIN1GRIN2B
SCHEMBL25888089 0.82 POLB (0.38) POLBGRIN1GRIN2BPTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018091389-A1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2018-05-24 WO disclosed