SCHEMBL20182759

SCHEMBL20182759

CCS(=O)(=O)c1cc(-c2ccc(C(F)(F)F)cc2)cnc1-c1nc2cc(C(F)(F)F)cnc2n1C

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.43
GRIN1 Q05586 3/20 0.35
GRIN2B Q13224 3/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
JAK3 P52333 1/20 0.35
DDR1 Q08345 3/20 0.35
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35
SCN9A Q15858 2/20 0.35
RORC P51449 1/20 0.34
CA12 O43570 1/20 0.34
CA9 Q16790 1/20 0.34
KCNH2 Q12809 1/20 0.34
MAPK10 P53779 1/20 0.34
PTGS2 P35354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30989728 0.90 POLB (0.39) POLBGRIN1GRIN2BALOX5APFEN1
SCHEMBL25885629 0.90 POLB (0.39) POLBGRIN1GRIN2BALOX5APFEN1
SCHEMBL14684583 0.90 POLB (0.48) POLBDDR1ALOX5APFEN1
SCHEMBL29360277 0.90 POLB (0.48) POLBDDR1ALOX5APFEN1
SCHEMBL25888089 0.89 POLB (0.38) POLBGRIN1GRIN2BMAPK10PTGS2
SCHEMBL20182758 0.89 POLB (0.44) POLBGRIN1GRIN2BDDR1ALOX5AP
SCHEMBL20182714 0.89 POLB (0.40) POLBGRIN1GRIN2BPTGS2
SCHEMBL17696196 0.88 PTGS2 (0.36) GRIN1GRIN2BJAK2JAK1TYK2
SCHEMBL18866344 0.87 POLB (0.42) POLBGRIN1GRIN2BDDR1PTGS2
SCHEMBL15868301 0.87 POLB (0.46) POLBDDR1ALOX5APFEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018091389-A1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2018-05-24 WO disclosed