SCHEMBL20184481

SCHEMBL20184481

CCC(=O)Nc1cccc(-c2nc(CC)nc3[nH]cc(C(=O)O)c23)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.48
CYP2D6 P10635 2/20 0.48
CYP2C19 P33261 2/20 0.48
TP53 P04637 4/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
USP2 O75604 1/20 0.48
CYP1A2 P05177 1/20 0.48
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
MAPK1 P28482 1/20 0.47
RAB9A P51151 4/20 0.46
NPC1 O15118 3/20 0.46
KDM4E B2RXH2 2/20 0.45
HSD17B10 Q99714 1/20 0.45
JAK3 P52333 9/20 0.44
HPGD P15428 1/20 0.44
POLB P06746 1/20 0.43
NR4A1 P22736 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20184594 0.90 JAK3 (0.43) MEN1KMT2AUSP2MAPTALDH1A1
SCHEMBL20184694 0.89 JAK3 (0.47) CYP3A4CYP2D6CYP2C19HSD17B10JAK3
SCHEMBL20184584 0.88 JAK3 (0.59) JAK3JAK2JAK1
SCHEMBL16245166 0.87 JAK3 (0.58) JAK3JAK2JAK1
SCHEMBL20184567 0.87 JAK3 (0.58) JAK3JAK2JAK1
SCHEMBL20184521 0.86 JAK3 (0.59) JAK3JAK2JAK1
SCHEMBL20184508 0.86 JAK3 (0.59) JAK3JAK2JAK1
SCHEMBL20184424 0.86 JAK3 (0.59) JAK3JAK2JAK1
SCHEMBL20184685 0.86 JAK3 (0.59) JAK3JAK2JAK1
SCHEMBL20184542 0.86 JAK3 (0.48) JAK3JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788000-B1 PYRROLOPYRIMIDINES AS JANUS KINASE INHIBITORS MERCK SHARP & DOHME (US) 2018-05-30 EP claimed