SCHEMBL20184694

SCHEMBL20184694

CCc1nc(-c2cccc(NC(=O)CC#N)c2)c2c(C(=O)O)c[nH]c2n1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 17/20 0.47
JAK2 O60674 5/20 0.47
BTK Q06187 1/20 0.44
HTT P42858 1/20 0.43
HSD17B10 Q99714 1/20 0.43
JAK1 P23458 3/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20184481 0.89 CYP3A4 (0.48) JAK3JAK2HSD17B10JAK1CYP3A4
SCHEMBL20184323 0.88 JAK3 (0.41) JAK3JAK2JAK1
SCHEMBL20184688 0.88 JAK3 (0.43) JAK3JAK2JAK1
SCHEMBL20184594 0.86 JAK3 (0.43) JAK3JAK2JAK1
SCHEMBL20184567 0.83 JAK3 (0.58) JAK3JAK2BTKJAK1
SCHEMBL16245166 0.83 JAK3 (0.58) JAK3JAK2JAK1
SCHEMBL20184429 0.83 JAK3 (0.54) JAK3JAK2JAK1
SCHEMBL20184677 0.82 F11 (0.43) JAK3JAK2
SCHEMBL20184584 0.82 JAK3 (0.59) JAK3JAK2JAK1
SCHEMBL20184508 0.82 JAK3 (0.59) JAK3JAK2JAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788000-B1 PYRROLOPYRIMIDINES AS JANUS KINASE INHIBITORS MERCK SHARP & DOHME (US) 2018-05-30 EP claimed