SCHEMBL20184516

SCHEMBL20184516

CCc1nc(-c2ccccc2F)c2c(C(=O)O)c[nH]c2n1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 5/20 0.52
JAK2 O60674 3/20 0.52
HSP90AB1 P08238 1/20 0.42
CHUK O15111 1/20 0.41
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
DHODH Q02127 6/20 0.37
ADORA2A P29274 2/20 0.37
ADORA1 P30542 2/20 0.37
ADORA3 P0DMS8 1/20 0.37
ADORA2B P29275 1/20 0.37
TACR3 P29371 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20184405 0.87 HSP90AB1 (0.45) JAK3JAK2HSP90AB1
SCHEMBL20184403 0.86 DHODH (0.42) JAK3JAK2HSP90AB1DHODH
SCHEMBL20184389 0.86 JAK3 (0.40) JAK3JAK2HSP90AB1CHUK
SCHEMBL20184670 0.85 HSP90AB1 (0.42) JAK3JAK2HSP90AB1CHUK
SCHEMBL20184525 0.84 JAK2 (0.49) JAK3JAK2CHUK
SCHEMBL20184489 0.82 JAK2 (0.51) JAK3JAK2DHODH
SCHEMBL20184555 0.81 HSP90AB1 (0.43) JAK3JAK2HSP90AB1CHUKDHODH
SCHEMBL20184360 0.80 JAK3 (0.60) JAK3HSP90AB1
SCHEMBL20184599 0.80 JAK3 (0.53) JAK3JAK2HSP90AB1CHUKDHODH
SCHEMBL20184528 0.79 JAK3 (0.41) JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788000-B1 PYRROLOPYRIMIDINES AS JANUS KINASE INHIBITORS MERCK SHARP & DOHME (US) 2018-05-30 EP claimed