SCHEMBL20184403

SCHEMBL20184403

CCc1nc(-c2ccccc2Cl)c2c(C(=O)O)c[nH]c2n1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.42
KMT2A Q03164 1/20 0.40
PRKAB2 O43741 3/20 0.38
PRKAG1 P54619 3/20 0.38
PRKAA2 P54646 3/20 0.38
PRKAA1 Q13131 3/20 0.38
PRKAG3 Q9UGI9 3/20 0.38
PRKAG2 Q9UGJ0 3/20 0.38
PRKAB1 Q9Y478 3/20 0.38
JAK2 O60674 3/20 0.38
JAK3 P52333 3/20 0.38
HPGD P15428 1/20 0.38
HSP90AB1 P08238 1/20 0.38
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
NR4A2 P43354 1/20 0.37
CNR1 P21554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20184405 0.87 HSP90AB1 (0.45) JAK2JAK3HSP90AB1RXRARXRB
SCHEMBL20184389 0.86 JAK3 (0.40) JAK2JAK3HSP90AB1
SCHEMBL20184516 0.86 JAK3 (0.52) DHODHJAK2JAK3HSP90AB1
SCHEMBL20184525 0.84 JAK2 (0.49) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL20184489 0.82 JAK2 (0.51) DHODHPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL20184700 0.81 JAK2 (0.40) DHODHPRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL20184478 0.80 JAK2 (0.53) DHODHJAK2JAK3
SCHEMBL20184672 0.78 JAK2 (0.54) DHODHKMT2AJAK2JAK3
SCHEMBL20184679 0.78 JAK3 (0.56) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL20184527 0.77 JAK2 (0.49) DHODHJAK2JAK3HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2788000-B1 PYRROLOPYRIMIDINES AS JANUS KINASE INHIBITORS MERCK SHARP & DOHME (US) 2018-05-30 EP claimed