SCHEMBL20187556

SCHEMBL20187556

F[C@@H](Br)Cc1ccc(Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.54
SLC6A2 P23975 2/20 0.50
SLC6A3 Q01959 2/20 0.50
IDO1 P14902 3/20 0.42
TAAR1 Q96RJ0 2/20 0.39
PPARG P37231 5/20 0.39
PPARA Q07869 5/20 0.39
LMNA P02545 1/20 0.38
CYP2A6 P11509 1/20 0.38
AGXT P21549 2/20 0.38
HTR2A P28223 1/20 0.35
HRH1 P35367 1/20 0.35
HTR2B P41595 1/20 0.35
CHRNA4 P43681 1/20 0.35
GAA P10253 1/20 0.35
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11566972 0.80 SLC6A4 (0.58) SLC6A4SLC6A2SLC6A3IDO1TAAR1
SCHEMBL1121849 0.78 TRPA1 (0.47) IDO1TAAR1LMNAAGXT
SCHEMBL2765367 0.78 SLC6A4 (0.56) SLC6A4SLC6A2SLC6A3IDO1TAAR1
SCHEMBL29092065 0.76 SLC6A4 (0.54) SLC6A4SLC6A2SLC6A3IDO1TAAR1
SCHEMBL28771419 0.76 SLC6A4 (0.54) SLC6A4SLC6A2SLC6A3IDO1TAAR1
SCHEMBL29091897 0.76 SLC6A4 (0.54) SLC6A4SLC6A2SLC6A3IDO1TAAR1
SCHEMBL4010409 0.76 SLC6A2 (0.61) SLC6A4SLC6A2SLC6A3IDO1TAAR1
SCHEMBL6425532 0.76 IDO1 (0.42) IDO1TAAR1PPARGPPARACYP2A6
SCHEMBL9481327 0.75 SLC6A4 (0.58) SLC6A4SLC6A2SLC6A3IDO1TAAR1
SCHEMBL459370 0.75 EPHX1 (0.50) SLC6A4SLC6A2SLC6A3TAAR1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3544979-A1 OXADIAZOLONES AS TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS H. Hoffnabb-La Roche Ag (CH) 2019-10-02 EP disclosed
WO-2018096159-A1 OXADIAZOLONES AS TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2018-05-31 WO disclosed