SCHEMBL20187646

SCHEMBL20187646

COc1cc2c(cc1OC)C(=O)c1oc(C(C)=O)cc1C2=O

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STAT3 P40763 5/20 0.64
ALDH1A1 P00352 2/20 0.64
LMNA P02545 1/20 0.44
RECQL P46063 1/20 0.44
PDE4A P27815 1/20 0.41
TNFSF11 O14788 1/20 0.41
CA9 Q16790 3/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CYP3A4 P08684 2/20 0.39
HTT P42858 1/20 0.39
MAPT P10636 2/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
LCK P06239 2/20 0.36
HPGD P15428 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20189157 0.82 STAT3 (0.66) STAT3ALDH1A1CA9CA1CA2
SCHEMBL20187637 0.82 STAT3 (0.66) STAT3ALDH1A1CA9CA1CA2
SCHEMBL20187669 0.82 STAT3 (0.57) STAT3ALDH1A1LMNARECQLCA9
SCHEMBL20187648 0.82 STAT3 (0.65) STAT3ALDH1A1LMNARECQLHTT
SCHEMBL20187658 0.80 STAT3 (0.58) STAT3ALDH1A1LMNARECQLCA9
Napabucasin SCHEMBL1883845 0.78 STAT3 (1.00) STAT3ALDH1A1LMNAHTTMAPT
SCHEMBL14656628 0.76 STAT3 (0.71) STAT3ALDH1A1LMNARECQLHTT
SCHEMBL14656586 0.76 STAT3 (0.71) STAT3ALDH1A1LMNARECQLHTT
SCHEMBL20191216 0.75 STAT3 (0.60) STAT3ALDH1A1LMNARECQLMAPT
SCHEMBL1882564 0.75 STAT3 (0.69) STAT3ALDH1A1LMNARECQLCA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018096401-A1 NEW NAPHTHO[2,3-B]FURAN DERIVATIVES BAN HITOSHI (JP) 2018-05-31 WO claimed
WO-2018096401-A1 NEW NAPHTHO[2,3-B]FURAN DERIVATIVES BAN HITOSHI (JP) 2018-05-31 WO disclosed