SCHEMBL20194159

SCHEMBL20194159

CC(C)C(=O)NC(=N)c1ccc(Cl)c(N)c1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.52
LMNA P02545 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
S1PR3 Q99500 10/20 0.42
S1PR4 O95977 3/20 0.42
S1PR1 P21453 2/20 0.42
S1PR5 Q9H228 2/20 0.42
NPC1 O15118 1/20 0.39
CASP3 P42574 1/20 0.39
RAB9A P51151 1/20 0.39
SENP8 Q96LD8 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39
HDAC1 Q13547 1/20 0.38
HPGD P15428 1/20 0.38
MAPK1 P28482 1/20 0.38
S1PR2 O95136 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20194125 0.84 GAA (0.41) KDM4EHPGD
SCHEMBL20194121 0.76 F2 (0.46) KDM4ELMNASMN1; SMN2S1PR3S1PR4
SCHEMBL20194127 0.75 S1PR3 (0.38) SMN1; SMN2S1PR3S1PR4S1PR1S1PR5
SCHEMBL5050812 0.72 NPC1 (0.56) KDM4ELMNASMN1; SMN2NPC1RAB9A
SCHEMBL21998506 0.71 ALDH1A1 (0.51) LMNASMN1; SMN2S1PR3S1PR4S1PR1
SCHEMBL7105778 0.70 PRKCI (0.56) KDM4ELMNASMN1; SMN2NPC1CASP3
SCHEMBL7913711 0.70 KDM4E (0.50) KDM4ELMNASMN1; SMN2NPC1CASP3
SCHEMBL20194149 0.70 CA12 (0.34) LMNAS1PR3S1PR4S1PR2
SCHEMBL312298 0.69 SRD5A2 (0.53) KDM4ELMNASMN1; SMN2NPC1RAB9A
SCHEMBL21099277 0.69 KDM4E (0.50) KDM4ELMNASMN1; SMN2NPC1CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3054955-B1 PYRROLOTRIAZINE KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-30 EP disclosed