SCHEMBL20194121

SCHEMBL20194121

CC(C)C(=O)NC(=N)c1cccc(N)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F2 P00734 1/20 0.46
PLG P00747 1/20 0.46
PRSS1 P07477 1/20 0.46
PRSS2 P07478 1/20 0.46
PRSS3 P35030 1/20 0.46
ALDH1A1 P00352 5/20 0.46
KDM4E B2RXH2 2/20 0.46
PBRM1 Q86U86 1/20 0.45
NPC1 O15118 2/20 0.43
MITF O75030 1/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
KDM4C Q9H3R0 1/20 0.42
ADRB2 P07550 2/20 0.42
ADRB1 P08588 2/20 0.42
ADRB3 P13945 2/20 0.42
MAPT P10636 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8302175 0.80 F2 (0.56) F2PLGPRSS1PRSS2PRSS3
SCHEMBL21998506 0.80 ALDH1A1 (0.51) ALDH1A1LMNAMAPTSMN1; SMN2NPSR1
SCHEMBL20194124 0.78 F2 (0.46) F2PLGPRSS1PRSS2PRSS3
SCHEMBL20194149 0.78 CA12 (0.34) ALDH1A1LMNAS1PR3S1PR2S1PR4
SCHEMBL20194126 0.77 SLC6A3 (0.36) ALDH1A1S1PR3RAB9AS1PR1
SCHEMBL20194127 0.77 S1PR3 (0.38) ALDH1A1MAPTSMN1; SMN2S1PR3S1PR2
SCHEMBL20194125 0.77 GAA (0.41) ALDH1A1KDM4EMAPTHSD17B10
SCHEMBL20194159 0.76 KDM4E (0.52) KDM4ENPC1LMNASMN1; SMN2S1PR3
SCHEMBL22649481 0.76 S1PR3 (0.40) ALDH1A1MAPTSMN1; SMN2HSD17B10S1PR3
SCHEMBL10401280 0.75 F2 (0.46) F2PLGPRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3054955-B1 PYRROLOTRIAZINE KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-30 EP disclosed