SCHEMBL20194149

SCHEMBL20194149

CC(C)C(=O)NC(=N)c1cc(N)cc(O)c1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA7 P43166 2/20 0.34
CA9 Q16790 2/20 0.34
CA14 Q9ULX7 2/20 0.34
ALDH1A1 P00352 3/20 0.33
CA5A P35218 1/20 0.32
GAA P10253 2/20 0.32
S1PR2 O95136 1/20 0.30
S1PR4 O95977 1/20 0.30
S1PR3 Q99500 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20194127 0.83 S1PR3 (0.38) ALDH1A1S1PR2S1PR4S1PR3
SCHEMBL20194126 0.83 SLC6A3 (0.36) ALDH1A1S1PR3
SCHEMBL20194121 0.78 F2 (0.46) ALDH1A1S1PR2S1PR4S1PR3LMNA
SCHEMBL20194125 0.74 GAA (0.41) CA12CA1CA2CA7CA9
SCHEMBL20194159 0.70 KDM4E (0.52) S1PR2S1PR4S1PR3LMNA
SCHEMBL21998506 0.69 ALDH1A1 (0.51) ALDH1A1GAAS1PR2S1PR4S1PR3
SCHEMBL30554535 0.67 CA12 (0.73) CA12CA1CA2CA7CA9
SCHEMBL1028307 0.67 CA12 (0.73) CA12CA1CA2CA7CA9
SCHEMBL30554557 0.67 CA12 (0.73) CA12CA1CA2CA7CA9
SCHEMBL6093793 0.66 PARP1 (0.50) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3054955-B1 PYRROLOTRIAZINE KINASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2018-05-30 EP disclosed