SCHEMBL20195393

SCHEMBL20195393

COCc1c(C2CC2)cccc1N(C)N

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTSR1 P30989 3/20 0.34
ADRA1A P35348 2/20 0.32
PDK2 Q15119 1/20 0.31
PDK4 Q16654 1/20 0.31
CYP1A2 P05177 1/20 0.31
HTR1A P08908 1/20 0.31
ADRA2A P08913 1/20 0.31
CYP2D6 P10635 1/20 0.31
THRB P10828 1/20 0.31
TSHR P16473 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
ADRA1D P25100 1/20 0.31
CYP2C19 P33261 1/20 0.31
ADRA1B P35368 1/20 0.31
THPO P40225 1/20 0.31
HSD17B10 Q99714 1/20 0.31
NISCH Q9Y2I1 1/20 0.31
GRM5 P41594 2/20 0.30
HTR2C P28335 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20686640 0.83 NOTUM (0.35) NTSR1
SCHEMBL18871241 0.81 PDK2 (0.33) PDK2PDK4HTR1A
SCHEMBL20342696 0.79 NOTUM (0.34) ADRA1APDK2PDK4CYP1A2CYP2D6
SCHEMBL18185030 0.78 ADRA1A (0.35) ADRA1APDK2PDK4CYP2D6CYP2C19
SCHEMBL20686851 0.77 MRGPRX4 (0.39) HTR1ATSHRLMNA
SCHEMBL22038794 0.77 HTR7 (0.44) ADRA1ACYP1A2HTR1AADRA2ACYP2D6
SCHEMBL20195514 0.76 HTR1A (0.39) ADRA1ACYP1A2HTR1AADRA2ACYP2D6
SCHEMBL19909901 0.76 AOC3 (0.31) CYP1A2CYP2D6TSHRHTR1DLMNA
SCHEMBL20686707 0.75 MRGPRX4 (0.41) CYP1A2HTR1ACYP2C19
SCHEMBL18871267 0.75 SLC22A12 (0.33) ADRA1ACYP1A2HTR1AADRA2ACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2990404-B1 TETRAZOLINONE COMPOUND AND USE OF SAME SUMITOMO CHEMICAL CO (JP) 2020-05-27 EP disclosed
EP-3029030-B1 TETRAZOLINONE COMPOUND, AND USE THEREFOR SUMITOMO CHEMICAL CO (JP) 2019-09-04 EP disclosed
EP-3029035-B1 TETRAZOLINONE COMPOUND, AND USE THEREOF SUMITOMO CHEMICAL CO (JP) 2018-05-30 EP disclosed