SCHEMBL20195482

SCHEMBL20195482

Cc1cccc(N(N)C(=O)N(C)N)c1COc1ccc(Br)nc1C

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
SLC22A12 Q96S37 1/20 0.34
PTGER1 P34995 1/20 0.32
SGMS2 Q8NHU3 1/20 0.32
BDKRB2 P30411 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22037708 0.85 HTR7 (0.42) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL20195553 0.85 ALDH1A1 (0.38) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL21317980 0.83 SLC22A12 (0.36) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL20686736 0.82 CYP1A2 (0.41) CYP1A2CYP2D6CYP2C19SLC22A12
SCHEMBL18831569 0.82 SLC22A12 (0.37) CYP1A2CYP2D6CYP2C19SLC22A12PTGER1
SCHEMBL21317966 0.81 SLC22A12 (0.40) CYP3A4CYP2C9CYP1A2CYP2D6CYP2C19
SCHEMBL18831565 0.80 SLC22A12 (0.39) SLC22A12
SCHEMBL18831320 0.79 F2 (0.36) SLC22A12
SCHEMBL22590904 0.79 LMNA (0.33) SLC22A12
SCHEMBL23506149 0.78 SLC22A12 (0.41) SLC22A12PTGER1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3029035-B1 TETRAZOLINONE COMPOUND, AND USE THEREOF SUMITOMO CHEMICAL CO (JP) 2018-05-30 EP disclosed