SCHEMBL2019635

SCHEMBL2019635

O=Cc1ccc(-c2ccc3c(c2)CNC3=O)s1

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PRF1 P14222 16/20 0.68
DAPK3 O43293 1/20 0.47
NTRK1 P04629 1/20 0.47
PIM1 P11309 1/20 0.47
FLT3 P36888 1/20 0.47
GSK3B P49841 1/20 0.47
ROCK1 Q13464 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
MAPT P10636 1/20 0.45
PGR P06401 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2020897 0.89 PRF1 (0.65) PRF1NTRK1FLT3GSK3BCLK4
SCHEMBL2020380 0.86 PRF1 (0.67) PRF1
SCHEMBL14761214 0.81 PRF1 (1.00) PRF1
SCHEMBL2042894 0.81 PRF1 (1.00) PRF1
SCHEMBL2042898 0.81 PRF1 (1.00) PRF1
SCHEMBL15570953 0.80 PRF1 (0.62) PRF1DAPK3NTRK1PIM1FLT3
SCHEMBL20923873 0.80 PRF1 (0.62) PRF1DAPK3NTRK1PIM1FLT3
SCHEMBL15571386 0.80 PRF1 (0.62) PRF1DAPK3NTRK1PIM1FLT3
SCHEMBL2054374 0.80 PRF1 (1.00) PRF1
SCHEMBL14761573 0.80 PRF1 (1.00) PRF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130065897-A1 COMPOUNDS, PREPARATION AND USES THEREOF PETER MACCALLUM CANCER INSTITUTE (AU) 2013-03-14 US disclosed
EP-2515903-A1 COMPOUNDS, PREPARATIONS AND USES THEREOF Peter MacCallum Cancer Institute (AU) 2012-10-31 EP disclosed
WO-2011075784-A1 COMPOUNDS, PREPARATIONS AND USES THEREOF PETER MACCALLUM CANCER INSTITUTE (AU) 2011-06-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130065897-A1 COMPOUNDS, PREPARATION AND USES THEREOF PRF1, GZMB, SERPINB1 PRF1 1/4885DAPK3 1267/4885NTRK1 4111/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.