SCHEMBL20196522

SCHEMBL20196522

CNc1ccc(CC(NC(=O)C(C)C(OC)C2CCCN2C)C(=O)OC)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.42
TSHR P16473 1/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
ALDH1A1 P00352 1/20 0.40
THRB P10828 1/20 0.40
HSD17B10 Q99714 1/20 0.40
ATM Q13315 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
IL2RA P01589 1/20 0.38
ALB P02768 1/20 0.38
IL2 P60568 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
POLB P06746 1/20 0.38
GFER P55789 1/20 0.38
DPP4 P27487 1/20 0.37
KMT2A Q03164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
YAP1 P46937 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18912329 0.89 GAA (0.54) GAATSHRCYP2C9CYP2C19ALDH1A1
SCHEMBL19647312 0.89 GAA (0.54) GAATSHRCYP2C9CYP2C19ALDH1A1
SCHEMBL22561427 0.87 KLKB1 (0.44) TSHRKMT2AMMP1
SCHEMBL22810961 0.82 POLB (0.49) GAAALDH1A1HSD17B10POLBKMT2A
SCHEMBL21699252 0.82 POLB (0.49) GAAALDH1A1HSD17B10POLBKMT2A
SCHEMBL15313443 0.82 POLB (0.49) GAAALDH1A1HSD17B10POLBKMT2A
SCHEMBL2734908 0.82 POLB (0.49) GAAALDH1A1HSD17B10POLBKMT2A
SCHEMBL9892967 0.82 POLB (0.49) GAAALDH1A1HSD17B10POLBKMT2A
SCHEMBL21781767 0.81 MMP13 (0.37)
SCHEMBL23209734 0.79 ATM (0.54) GAACYP2C9CYP2C19ALDH1A1THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3327027-A1 CYTOTOXIC PEPTIDES AND ANTIBODY DRUG CONJUGATES THEREOF Pfizer Inc (US) 2018-05-30 EP disclosed