SCHEMBL20197443

SCHEMBL20197443

[O-][S+](Nc1ccc(-c2csc(-c3csc4ccccc34)n2)c(Cl)c1)C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
C1S P09871 1/20 0.39
CYP1A1 P04798 4/20 0.37
CYP1B1 Q16678 4/20 0.37
CYP1A2 P05177 3/20 0.37
CYP19A1 P11511 1/20 0.36
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TEK Q02763 1/20 0.34
AMY1A P0DUB6 1/20 0.34
EGFR P00533 2/20 0.33
KDM4E B2RXH2 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
EIF4E P06730 2/20 0.33
PGK1 P00558 1/20 0.32
IGF1R P08069 1/20 0.32
SRC P12931 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20197337 0.84 CYP1A2 (0.40) C1SCYP1A1CYP1B1CYP1A2CYP19A1
SCHEMBL16535825 0.81 KDM1A (0.39) C1SCYP1A1CYP1B1CYP1A2CYP19A1
SCHEMBL20197238 0.80 CYP19A1 (0.44) CYP19A1AMY1AKDM4ENPC1RAB9A
SCHEMBL20197304 0.78 CDK2 (0.39) C1SCYP1A1CYP1B1CYP1A2CYP19A1
SCHEMBL20197479 0.78 EIF4E (0.39) CYP1A2MAPTKDM4ENPC1RAB9A
SCHEMBL20197235 0.76 SREBF2 (0.42) MAPTKDM4E
SCHEMBL20197481 0.76 EIF4E (0.37) KDM4ENPC1RAB9ASMN1; SMN2CRHBP
SCHEMBL20197159 0.76 CYP19A1 (0.33) CYP1A1CYP1B1CYP1A2CYP19A1AMY1A
SCHEMBL20197301 0.74 KDM4E (0.34) C1SCYP19A1MAPTKDM4ENPC1
SCHEMBL20197223 0.74 SREBF2 (0.42) MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3038622-B1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECH LLC (US) 2018-05-30 EP disclosed