SCHEMBL20199981

SCHEMBL20199981

COC(=O)CN1CCN(CC(=O)OC)CCN(CC(=O)N(CC(=O)O)c2ccccc2)CCN(CC(=O)OC)CC1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.43
CACNA1C Q13936 3/20 0.43
CACNA2D1 P54289 2/20 0.43
CACNA1B Q00975 2/20 0.43
CACNB1 Q02641 2/20 0.43
ALDH1A1 P00352 3/20 0.42
OPRM1 P35372 4/20 0.41
SIGMAR1 Q99720 3/20 0.41
KDM4E B2RXH2 2/20 0.40
TSHR P16473 2/20 0.40
AURKA O14965 1/20 0.39
TACR1 P25103 1/20 0.39
MLYCD O95822 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20187534 0.86 CACNA2D1 (0.49) DRD4CACNA1CCACNA2D1CACNA1BCACNB1
SCHEMBL20187617 0.81 CACNA2D1 (0.45) DRD4CACNA1CCACNA2D1CACNA1BCACNB1
SCHEMBL20199872 0.80 DRD4 (0.42) DRD4CACNA1CCACNA2D1CACNA1BCACNB1
SCHEMBL20199982 0.80 ALDH1A1 (0.46) DRD4ALDH1A1OPRM1SIGMAR1TACR1
SCHEMBL22112586 0.80 ALDH1A1 (0.47) ALDH1A1
SCHEMBL1387733 0.78 ALDH1A1 (0.43) DRD4CACNA1CCACNA2D1CACNA1BCACNB1
SCHEMBL22403100 0.78 CACNA2D1 (0.45) DRD4CACNA1CCACNA2D1CACNA1BCACNB1
SCHEMBL1387794 0.77 MEN1 (0.42) CACNA1CCACNA2D1CACNA1BCACNB1ALDH1A1
SCHEMBL9080067 0.76 ALDH1A1 (0.42) DRD4CACNA1CCACNA2D1CACNA1BCACNB1
SCHEMBL20200052 0.76 ALDH1A1 (0.37) DRD4ALDH1A1OPRM1SIGMAR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018096082-A1 HIGH RELAXIVITY GADOLINIUM CHELATE COMPOUNDS FOR USE IN MAGNETIC RESONANCE IMAGING BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-05-31 WO disclosed