SCHEMBL1387733

SCHEMBL1387733

O=C(O)CN1CCN(CC(=O)O)CCN(CC(=O)N(CC(=O)O)c2ccc(-c3ccccc3)cc2)CCN(CC(=O)O)CC1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
TSHR P16473 2/20 0.43
CACNA2D1 P54289 2/20 0.42
CACNA1B Q00975 2/20 0.42
CACNB1 Q02641 2/20 0.42
CACNA1C Q13936 2/20 0.42
LMNA P02545 3/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
DRD4 P21917 1/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
GAA P10253 1/20 0.38
MLYCD O95822 1/20 0.38
TP53 P04637 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PDE4B Q07343 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9080067 0.97 ALDH1A1 (0.42) ALDH1A1KDM4ETSHRCACNA2D1CACNA1B
SCHEMBL20187534 0.91 CACNA2D1 (0.49) ALDH1A1KDM4ETSHRCACNA2D1CACNA1B
SCHEMBL1387794 0.84 MEN1 (0.42) ALDH1A1KDM4ETSHRCACNA2D1CACNA1B
SCHEMBL22403100 0.83 CACNA2D1 (0.45) ALDH1A1KDM4ETSHRCACNA2D1CACNA1B
SCHEMBL9079952 0.81 MLYCD (0.40) ALDH1A1KDM4ETSHRLMNADRD4
SCHEMBL20187617 0.81 CACNA2D1 (0.45) ALDH1A1KDM4ETSHRCACNA2D1CACNA1B
Tromethamine SCHEMBL9264448 0.79 GSTO1 (0.38) ALDH1A1KDM4ETSHRLMNANPC1
SCHEMBL20199981 0.78 DRD4 (0.43) ALDH1A1KDM4ETSHRCACNA2D1CACNA1B
SCHEMBL1387857 0.78 ALDH1A1 (0.43) ALDH1A1LMNANPC1SMN1; SMN2
SCHEMBL9080745 0.78 GSTO1 (0.40) ALDH1A1KDM4ETSHRCACNA2D1CACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-H08511809-A 1996-12-10 JP claimed
US-5573752-A Aromatic amide compounds and metal chelates thereof BRACCO INTERNATIONAL B.V. 1996-11-12 US claimed
EP-0702677-A1 AROMATIC AMIDE COMPOUNDS AND METAL CHELATES THEREOF BRACCO International B.V. (NL) 1996-03-27 EP claimed
WO-1995027705-A1 AROMATIC AMIDE COMPOUNDS AND METAL CHELATES THEREOF BRACCO INTERNATIONAL B.V. (NL) 1995-10-19 WO claimed
US-5573752-A Aromatic amide compounds and metal chelates thereof BRACCO INTERNATIONAL B.V. 1996-11-12 US disclosed
WO-1995027705-A1 AROMATIC AMIDE COMPOUNDS AND METAL CHELATES THEREOF BRACCO INTERNATIONAL B.V. (NL) 1995-10-19 WO disclosed