SCHEMBL20203564

SCHEMBL20203564

CC(C)c1ccc2c(n1)CCN(C(=O)[C@H]1C[C@@H](O)CN1CC(C)c1ccc3c(n1)CCN(C(=O)[C@@H]1CCCNC1)C3)C2

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TYRO3 Q06418 2/20 0.34
GABRG2 P18507 3/20 0.33
GABRB3 P28472 3/20 0.33
GABRA5 P31644 3/20 0.33
PARP1 P09874 1/20 0.32
CDK4 P11802 1/20 0.31
CDK2 P24941 1/20 0.31
CDK6 Q00534 1/20 0.31
HDAC6 Q9UBN7 2/20 0.31
KCNH2 Q12809 1/20 0.31
KEAP1 Q14145 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23733451 0.85 KEAP1 (0.40) TYRO3GABRG2GABRB3GABRA5PARP1
SCHEMBL20203531 0.80 TLR9 (0.41) GABRG2GABRB3GABRA5PARP1CDK4
SCHEMBL20203599 0.76 CDK4 (0.36) CDK4CDK2CDK6
SCHEMBL23733483 0.75 CDK4 (0.35) GABRG2GABRB3GABRA5CDK4CDK2
SCHEMBL20203431 0.74 KEAP1 (0.41) GABRG2GABRB3GABRA5CDK4HDAC6
SCHEMBL21414410 0.73 KEAP1 (0.43) GABRG2GABRB3GABRA5PARP1HDAC6
SCHEMBL20203643 0.72 HSP90AA1 (0.40) GABRG2GABRB3GABRA5CDK4CDK2
SCHEMBL23733474 0.71 CDK1 (0.45) PARP1CDK4CDK2CDK6
SCHEMBL20203529 0.71 CDK1 (0.45) PARP1CDK4CDK2CDK6
SCHEMBL20203457 0.70 GRM5 (0.49) GABRG2GABRB3GABRA5CDK4HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018097297-A1 PYRIDO[3, 4-D]PYRIMIDINE DERIVATIVE AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF 帝人ファーマ株式会社 2018-05-31 WO disclosed